TG100-115 Cas 677297-51-7 PI3K Inhibitors
TG100-115 Cas 677297-51-7 PI3K Inhibitors
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Chemical Information
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Product name:TG100-115 |
Purity:98% min |
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CAS NO:677297-51-7 |
Solubility:DMSO5.45 mg/mL (15.74 mM) |
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Molecular Formula:C18H14N6O2 |
Package:Package according to customer requirements |
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Molecular Weight:346.343 |
Storage:Store at -20℃ |
Quality control
Remarks
TG100-115, inhibited PI3K and -(IC50 values of 83 and 235 nM, respectively), whereas both PI3K and - were relatively unaffected (IC50 values>1 M). As a gauge of general specificity, TG100-115 was also assayed against a 133 protein kinase panel, none of which was inhibited at IC50 values <1 M.
Related Products:
Idelalisib; Almorexant HCL; IC-87114; Pictilisib; Pictilisib mesylate; XL147; PIK-90; Omipalisib; Buparlisib;A66; AS-252424; GSK2636771; CH5132799; 3-methyladenine; AS-604850
References
[1].Doukas J, et al. Phosphoinositide 3-kinase gamma/delta inhibition limits infarct size after myocardial ischemia/reperfusion injury. Proc Natl Acad Sci U S A. 2006 Dec 26;103(52):19866-71.
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