Synthesis Inhibitors
Tenovin-6 cas 1011557-82-6
Chemical Information Product name:Tenovin-6 Purity:98% min CAS NO:1011557-82-6 Solubility:DMSO : ≥ 31 mg/mL (68.19 mM) Molecular Formula:C25H34N4O2S Package:Package according to customer requirements Molecular Weight:454.628 Storage:Store at -20℃ Remarks Tenovin-6, also known as Tnv-6, is a bioactive small molecule SIRT2 inhibitor with anti-neoplastic activity. Inhibition of the Sirtuin class of protein deacetylases with activation of p53 function is associated with the pro
Zolmitriptan cas 139264-17-8
Chemical Information Product name:Zolmitriptan Purity:98% min CAS NO:139264-17-8 Solubility:DMSO: 58 mg/mL (201.83 mM) Molecular Formula:C16H21N3O2 Package:Package according to customer requirements Molecular Weight:287.357 Storage:Store at -20℃ Remarks Zolmitriptan is a member of the triptan class agents with anti-migraine property. Zolmitriptan selectively binds to and activates serotonin (5-HT) 1B expressed in intracranial arteries and 5_HT 1D receptors located on
Dimethyl 3-(3-chlorophenoxy)-2-oxopropylphosphonate cas 40665-94-9
Chemical Information Product name:Dimethyl 3-(3-chlorophenoxy)-2-oxopropylphosphonate Purity:98% min CAS NO:40665-94-9 Solubility: Molecular Formula:C11H14ClO5P Package:Package according to customer requirements Molecular Weight:292.653 Storage:Store at -20℃ Remarks Synonyms: DIMETHYL 3-(3-CHLOROPHENOXY)-2-OXOPROPYLPHOSPHONATE; Dimethyl 3-(3-chlorophenoxy)-2-oxopropylphosphonate, 98 %; 3-(m-Chlorophenoxy)-2-oxopropylphosphonic acid dimethyl ester; [2-Oxo-3-(3-chloro-phenoxy)
sitafloxacin Hydrate cas 163253-35-8
Chemical Information Product name:Sitafloxacin Hydrate Purity:98% min CAS NO:163253-35-8 Solubility:DMSO : 8.9 mg/mL (20.37 mM) Molecular Formula:C19H20ClF2N3O4 Package:Packaging according to customer requirements. Molecular Weight:427.83 Storage:Store at -20℃ Quality control COA Remarks Sitafloxacin is a new-generation, broad-spectrum oral fluoroquinolone that is very active against many Gram-positive, Gram-negative and anaerobic clinical isolates, including strains
Cerivastatin cas 145599-86-6
Name Cerivastatin CAS NO. 145599-86-6 Molecular Formula C26H33FNNaO5 Molecular Weight 481.53 Standard Assay ≥99% Structure Remarks Order None of the products will be supplied to countries in which this could be in conflict with the existing patents. However the final responsibility lies with the Buyer.
AT9283 cas 896466-04-9
Chemical Information Product name:AT9283 Purity:98% min CAS NO:896466-04-9 Solubility:DMSO : ≥ 100 mg/mL (262.17 mM) Molecular Formula:C19H23N7O2 Package:Package according to customer requirements Molecular Weight:381.432 Storage:Store at -20℃ Quality control COA Remarks AT9283 is a multikinase inhibitor, is also a small-molecule inhibitor of several kinases with potential antineoplastic activity. Multikinase inhibitor AT9283 binds to and inhibits Aurora kinases A and B, JAK2
sitafloxacin isomer I(SSR) cas 127254-11-9
Chemical Information Product name:sitafloxacin isomer I(SSR) Purity:98% min CAS NO:127254-11-9 Solubility:DMSO Molecular Formula:C19H18ClF2N3O3 Package:Package according to customer requirements Molecular Weight:409.814 Storage:Store at -20℃ Remarks Properties: Density: 1.63 Boiling Point: 629.221ºC at 760 mmHg Related Prodcuts: sitafloxacin isomer II(RSR); sitafloxacin isomer III(RRS); Sitafloxacin Hydrate
sitafloxacin isomer III(RRS) cas 127254-10-8
Chemical Information Product name:sitafloxacin isomer III(RRS) Purity:98% min CAS NO:127254-10-8 Solubility:DMSO Molecular Formula:C19H18ClF2N3O3 Package:Package according to customer requirements Molecular Weight:409.814 Storage:Store at -20℃ Remarks Properties: Density: 1.63 g/cm3 Boiling Point: 629.2ºC at 760 mmHg Flash Point: 334.3ºC Related Prodcuts: sitafloxacin isomer I(SSR); sitafloxacin isomer II(RSR); Sitafloxacin Hydrate
Rigosertib sodium salt cas 1225497-78-8
Chemical Information Product name:Rigosertib sodium salt Purity:98% min CAS NO:1225497-78-8 Solubility:H2O : ≥ 52 mg/mL (109.83 mM) Molecular Formula:C21H24NNaO8S Package:Package according to customer requirements Molecular Weight:473.472 Storage:Store at -20℃ Remarks Rigosertib (ON-01910 sodium salt) is a synthetic benzyl styryl sulfone analogue with potential antineoplastic activity. Polo-like kinase 1 inhibitor ON 01910.Na inhibits polo-like kinase1 (Plk1), inducing
TPX-0046
Chemical Information Product name:TPX-0046 Purity:CR3939 CAS NO:TPX-0046 Solubility:Soluble in DMSO Molecular Formula: Package:Package according to customer requirements Molecular Weight: Storage:Store at -20℃ Remarks TPX-0046 is a novel and potent RET/SRC inhibitor for RET-driven cancers. References https://www.sciencedirect.com/science/article/pii/S0923753419587282
Dibenzosuberone cas 1210-35-1
Chemical Information Product name:Dibenzosuberone Purity:98% min CAS NO:1210-35-1 Solubility:Soluble in DMSO Molecular Formula:C15H12O Package:Package according to customer requirements. Molecular Weight:208.255 Storage:-20ºC Remarks Amitriptyline impurity, a potential antidepressant compound. Synonyms: 5,6-dihydrodibenzo[2,1-b:2',1'-f][7]annulen-11-one; 5H-Dibenzo[a,d]cyclohepten-5-one, 10,11-dihydro-; Properties: Appearance & Physical State: Clear to yellow liquid Density:
TPX-0131
Chemical Information Product name:TPX-0131 Purity:99.0% min CAS NO:TPX-0131 Solubility:Soluble in DMSO Molecular Formula: Package:Package according to customer requirements Molecular Weight: Storage:Store at -20℃ Remarks ALK inhibitor TPX-0131
sitafloxacin isomer II(RSR) cas 1271199-06-8
Chemical Information Product name:sitafloxacin isomer II(RSR) Purity:98% min CAS NO:1271199-06-8 Solubility:Soluble in DMSO Molecular Formula: Package:Package according to customer requirements Molecular Weight: Storage:Store at -20℃ Remarks sitafloxacin isomer II(RSR) cas 1271199-06-8 Related Prodcuts: sitafloxacin isomer I(SSR); sitafloxacin isomer III(RRS); Sitafloxacin Hydrate
Prostacyclin sodium salt Epoprostenol sodium cas 61849-14-7
Chemical Information Product name:Prostacyclin sodium salt Epoprostenol sodium Purity:98% min CAS NO:61849-14-7 Solubility:Soluble in DMSO, not in water Molecular Formula:C20H31NaO5 Package:Package according to customer requirements Molecular Weight:374.45 Storage:Store at -20℃ Remarks Epoprostenol sodium (Prostaglandin I2 (sodium salt)), the synthetic form of the natural prostaglandin derivative prostacyclin (prostaglandin I2), is registered worldwide for the treatment of
(E)-3-(4-amino-3,5-dimethylphenyl)acrylonitrile cas 500292-94-4
Chemical Information Product name:(E)-3-(4-amino-3,5-dimethylphenyl)acrylonitrile Purity:98% min CAS NO:500292-94-4 Solubility:Soluble in DMSO Molecular Formula:C11H12N2 Package:Package according to customer requirements. Molecular Weight:172.226 Storage:-20ºC Remarks Synonyms: (E)-3-(4-amino-3,5-dimethylphenyl)acrylonitrile; (E)-3-(4-amino-3,5-dimethylphenyl)acrylonitrile HCl; -3-(4-Amino-3,5-dimethylphenyl); 2-Propenenitrile, 3-(4-aMino-3,5-diMethylphenyl)-, (2E)-; (2E)-3-
Limaprost Alfadex N-2 cas 94924-48-8
Chemical Information Product name:Limaprost Alfadex N-2 Purity:98% min CAS NO:94924-48-8 Solubility:Soluble in DMSO Molecular Formula:C35H64O5Si2 Package:Packaging according to customer requirements Molecular Weight:623.06 Storage:Store at -20℃ Quality control COA Remarks Limaprost INTERMEDIATE CAS NO:94924-48-8 , 98% min Chemical Name: methyl (E)-7-((1R,2R,3R)-3-((tert-butyldimethylsilyl)oxy)-2-((3S,5S,E)-3-((tert-butyldimethylsilyl)oxy)-5-methylnon-1-en-1-yl)-5-oxocyclopent
TPX-0022 CSF1R-IN-2 cas 2271119-26-5
Chemical Information Product name:TPX-0022 CSF1R-IN-2 Purity:98.0% min CAS NO:2271119-26-5 Solubility:DMSO : 25 mg/mL (61.06 mM; Need ultrasonic) Molecular Formula:C20H20FN7O2 Package:Package according to customer requirements Molecular Weight:409.42 Storage:Store at -20℃ Remarks TPX-0022, also known as CSF1R-IN-2, is an orally bioavailable multi-targeted kinase inhibitor with a novel three-dimensional macrocyclic structure that inhibits the MET, CSF1R (colony stimulating
CC-401 cas 395104-30-0
Chemical Information Product name:CC-401 Purity:98% min CAS NO:395104-30-0 Solubility: Molecular Formula:C22H24N6O Package:Package according to customer requirements Molecular Weight:388.466 Storage:Store at -20℃ Remarks CC-401 is a second generation ATP-competitive anthrapyrazolone c-Jun N terminal kinase (JNK) inhibitor with potential antineoplastic activity. Based on the chemistry of SP600125, another anthrapyrazolone inhibitor of JNK, CC-401 competitively binds the ATP
Sitaxsentan sodium cas 210421-74-2
Chemical Information Product name:Sitaxsentan sodium Purity:98% min CAS NO:210421-74-2 Solubility:DMSO : 100 mg/mL (209.69 mM) Molecular Formula:C18H14ClN2NaO6S2 Package:Packaging according to customer requirements. Molecular Weight:476.89 Storage:Store at -20℃ Quality control COA Remarks Sitaxentan, also known as TBC-11251 and IPI 1040, is a medication for the treatment of pulmonary arterial hypertension (PAH). It was marketed as Thelin. In 2010, Pfizer voluntarily removed
Imidazole ketone erastin (PUN30119) cas 1801530-11-9
Chemical Information Product name:Imidazole ketone erastin (PUN30119) Purity:98.0% min CAS NO:1801530-11-9 Solubility:DMSO: 100 mg/mL (152.63 mM) Molecular Formula:C35H35ClN6O5 Package:Package according to customer requirements. Molecular Weight:655.14 Storage:2-8°C Remarks Imidazole ketone erastin (PUN30119, IKE) is a potent, selective, and metabolically stable system xc– inhibitor and inducer of ferroptosis. Chemical Properties Boiling point: 886.5±75.0 °C(Predicted)