Taizhou Crene Biotechnology Co., Ltd.
                                                                                                           
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Chemicals Chemical Reagents

KGA-2727 cas 666842-36-0

Price Negotiable
Price: Negotiable
MOQ: 1g
Delivery Time: Negotiable
Brand: Crene
Product Description
Chemical Information
Product name:KGA-2727 Purity:98.0% min
CAS NO:666842-36-0 Solubility:DMSO : 100 mg/mL (186.35 mM; Need ultrasonic)
Molecular Formula:C26H40N4O8 Package:Package according to customer requirements
Molecular Weight:536.63 Storage:Store at -20℃
Remarks

KGA-2727 is a potent, selective, high-affinity inhibitor of sodium glucose cotransporter 1 (SGLT1) with Ki of 97.4 nM and 43.5 nM for human SGLT1 and rat SGLT1, respectively. The selectivity ratios (Ki for SGLT2/Ki for SGLT1) of KGA-2727 are 140 (human) and 390 (rat). KGA-2727 exhibits antidiabetic efficacy in rodent models.

 

Properties:

Boiling point: 839.6±65.0 °C(Predicted)

density: 1.308±0.06 g/cm3(Predicted)

pka: 12.65±0.70(Predicted)

 

 

 

SGLT Inhibitors Related Prodcuts:

Canagliflozin; Empagliflozin; Sotagliflozin; Ertugliflozin; Dapagliflozin

References
[1] Shibazaki T, et al. J Pharmacol Exp Ther. 2012 Aug;342(2):28

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Company Taizhou Crene Biotechnology Co., Ltd.
Location Add: Economic Developed Zone of Taizhou Zhejiang China.

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